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Mots clés : Targeted cancer therapies, Antibody-Drug Conjugates

Publications


Selective Protein (Post-)modifications through Dynamic Covalent Chemistry: Self-activated SAr Reactions.

Esteve F, Schmitt JL, Kolodych S, Koniev O, Lehn JM

J Am Chem Soc. 2025 01 2;:

Antibody-Vincristine Conjugates as Potent Anticancer Therapeutic Agents.

Boos A, Most J, Cahuzac H, Moreira da Silva L, Daubeuf F, Erb S, Cianférani S, Hernandez-Alba O, Semenchenko C, Dovgan I, Kolodych S, Detappe A, Dantzer F, Wagner A, Zeniou M, Chaubet G

J Med Chem. 2024 12 16;:

INA03, a potent transferrin-competitive antibody-drug conjugate against CD71, for a safer acute leukemia treatment.

Bratti M, Stubbs E, Kolodych S, Souchet H, Kelly L, Merlin J, Marchal M, Castellano R, Josselin E, Pasquer H, Benajiba L, Puissant A, Koniev O, Collette Y, Belanger C, Hermine O, Monteiro RC, Launay P

Mol Cancer Ther. 2024 04 20;:

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