Nightmares and hallucinations with aprepitant and opium powder: a suspected drug-drug interaction.

Fiche publication


Date publication

novembre 2018

Journal

British journal of clinical pharmacology

Auteurs

Membres identifiés du Cancéropôle Est :
Pr BOUCHE Olivier


Tous les auteurs :
Narjoux G, Clarenne J, Azzouz B, Zeller PS, Slimano F, Bouché O

Résumé

Polypharmacy of elderly oncology patients and fragmented medication management are well-known risk factors for drug-drug interactions (DDIs). These interactions can occur among antineoplastic, ongoing chronic treatment(s) and chemotherapy-associated treatments, like antiemetics. Clinically relevant interactions based on enzyme- or transporter-inhibition phenomena of active drugs can increase the frequency of their DDIs. We describe a strongly suspected elderly cancer patient's DDI between aprepitant and opium powder in the context of an irinotecan-based regimen manifested by nightmares and visual hallucinations. We discuss this DDI's hypothetical pharmacological mechanisms and management.

Mots clés

OCT1, UGT2B7, aprepitant, drug-drug interaction, irinotecan, opium powder

Référence

Br J Clin Pharmacol. 2018 Nov 26;: