o-Nitrobenzyl photoremovable groups with fluorescence uncaging reporting properties.

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Date publication

août 2018

Journal

Organic & biomolecular chemistry

Auteurs

Membres identifiés du Cancéropôle Est :
Dr SPECHT Alexandre


Tous les auteurs :
Abou Nakad E, Bolze F, Specht A

Résumé

o-Nitrobenzyl (o-NB) derivatives are the most widely applied photoremovable groups for the study of dynamic biological processes. By introducing different substituents to the benzylic position we were able to generate a fluorescence signal upon irradiation. This signal originates from the formation of a nitrosoketone by-product able to achieve a keto-enol tautomerism leading to pi-conjugated α-hydroxystilbene derivatives. These o-NB caging groups can be used to directly monitor the uncaging event by the release of a detectable fluorescent side-product.

Référence

Org. Biomol. Chem.. 2018 08 22;16(33):6115-6122