Harnessing medically relevant metals onto water-soluble subphthalocyanines: towards bimodal imaging and theranostics.

Fiche publication


Date publication

février 2015

Journal

Dalton transactions (Cambridge, England : 2003)

Auteurs

Membres identifiés du Cancéropôle Est :
Dr DECREAU Richard, Pr PERRIER-CORNET Jean-Marie


Tous les auteurs :
Bernhard Y, Winckler P, Perrier-Cornet JM, Decréau RA

Résumé

Subphthalocyanine (SubPc), a putative fluorophore for optical imaging (OI), was conjugated to chelating ligands (DOTA, DTPA) affording water-soluble conjugates complexed with (non-radioactive) metals relevant to the following medical imaging techniques/therapies: MRI (Gd), PET (Cu, Ga), SPECT (In, Ga, Lu), RIT (Cu, Lu, Y), and NCT (Gd). Magneto-optical properties of ditopic gadolinium species (and optical properties of other metal containing species) were examined (brightness (ε × ΦF) and relaxivity R1) and fluorescence confocal/biphoton microscopy studies were conducted.

Mots clés

Cell Line, Tumor, Cell Survival, drug effects, Humans, Indoles, chemistry, Magnetic Resonance Spectroscopy, methods, Melanoma, Experimental, chemistry, Metals, chemistry, Solubility, Water, chemistry

Référence

Dalton Trans. 2015 Feb 21;44(7):3200-8