Highly Recyclable Self-Supported Chiral Catalysts for the Enantioselective alpha-Hydrazination of beta-Ketoesters.

Fiche publication


Date publication

octobre 2013

Auteurs

Membres identifiés du Cancéropôle Est :
Dr BELLEMIN-LAPONNAZ Stéphane


Tous les auteurs :
Torres M, Maisse-Francois A, Bellemin-Laponnaz S

Résumé

Multitopic chiral copper complexes based on bis(oxazoline) have been applied in the enantioselective -hydrazination of -ketoesters. High yields and excellent enantioselectivities were obtained. Furthermore, the catalytic systems have been recovered in up to ten cycles without loss of activity or enantioselectivity. The formation of coordination polymers [polytopic ligand-Cu](n) has been confirmed by UV/Vis titrations. Significant metal leaching was observed on increasing the topicity of the ligand. The nature of the catalyst was studied by nonlinear effect experiments.

Référence

Chemcatchem. 2013 Oct;5(10):3078-85.