Photochemical aryl radical cyclizations to give (E)-3-ylideneoxindoles.

Fiche publication


Date publication

janvier 2014

Auteurs

Membres identifiés du Cancéropôle Est :
Pr SAPI Janos, Dr GERARD Stéphane


Tous les auteurs :
Gurry M, Allart-Simon I, McArdle P, Gerard S, Sapi J, Aldabbagh F

Résumé

(E)-3-Ylideneoxindoles are prepared in methanol in reasonable to good yields, as adducts of photochemical 5-exo-trig of aryl radicals, in contrast to previously reported analogous radical cyclizations initiated by tris(trimethylsilyl)silane and azo-initiators that gave reduced oxindole adducts.

Référence

Molecules. 2014 Sep 30;19(10):15891-9